Shanghai Sonyt Biotechnology Co., Ltd. yog ib qho ntawm cov ua lag luam thiab cov muag khoom ntawm selepessin acetate hauv Suav teb, kuj txhawb kev pabcuam kev cai. Txais tos rau kev lag luam wholesale bulk zoo selepessin acetate los ntawm peb lub hoobkas. Tiv tauj peb kom paub meej ntxiv.
| Khoom npe | Selepessin acetate hmoov |
| Kev piav qhia | Selepressin yog ib qho tshiab - tiam neeg xaiv vasopressin V1a receptor agonist. Nws tshwj xeeb khi rau V1a receptors ntawm vascular du leeg, muaj zog constricts peripheral cov hlab ntsha thiab ua rau kom cov hlab ntsha siab, siv rau kev tshawb fawb kev kho mob hauv vasodilatory shock. Piv nrog cov neeg vasopressin, optimized los ntawm cov amino acid ib ntus, nws nyuam qhuav qhib V2 receptors, tsis txhob muaj kev phiv xws li dej thiab sodium retention thiab antidiuresis, nrog rau cov kev xaiv ntau dua. Nws yog ib qho tshiab - tiam tshiab peptide rau septic shock, vasodilatory hypotension, cardiovascular pharmacology thiab vasopressin receptor function research. |
| Peptide Purity (HPLC, %) | 95% / 98% / 99% |
| Dawb peptide molecular mis | C₄₆H₆₅N₁₅O₁₂S₂ |
| Dawb peptide molecular hnyav (Da) | 1088.24, siab dua rau daim ntawv acetate |
| Hom qauv | Hloov kho cyclic nonapeptide, ib khub ntawm intramolecular disulfide daim ntawv cog lus, qhov chaw- hloov kho los txhim kho V1a xaiv, acetate ntsev |
Product Basic Information Table
| Khoom Lub Npe Lus Askiv | Product Abbreviation / Alias | Function Tags (comma-sib cais) | Core Structure | Molecular Formula | Exact Mass (Da) | Qhov nruab nrab MW (Da) | Daim ntawv ntsev | Ntev (aa) |
| Selepessin acetate hmoov | TIAB SA 202158 | Muaj kev xaiv V1a receptor agonist, pressor & anti- poob siab, tsis muaj V2 antidiuretic phiv | Hloov kho cyclic nonapeptide nrog ib daim ntawv cog lus intramolecular disulfide kom muaj kev sib haum xeeb; multi-site amino acid hloov kho tau zoo txhim kho V1a receptor selectivity nrog yuav luag tsis muaj V2 receptor-cov dej nruab nrab-sodium retention kev ua | Dawb puag: C₄₆H₆₅N₁₅O₁₂S₂; Daim ntawv ntsev: C₄₆H₆₅N₁₅O₁₂S₂·xC₂H₄O₂ | 1087.44 | 1088.24 | Acetate | 9 |
Physicochemical Solubility & Cia Parameters
| Khoom Code | Qhov tshwm sim | Ntev - Lub Sij Hawm Cia | Luv - Lub Sij Hawm Cia | Kev daws teeb meem | Khoom hmoov ruaj khov |
| PEB-SEL001 | hmoov dawb | Khaws ntawm -20 degree, kaw, qhuav thiab tiv thaiv los ntawm lub teeb. Aliquot rau cia. Tsis txhob muaj cov tshuaj tiv thaiv muaj zog thiab rov ua kom khov-thaw mus ntxiv. | ruaj khov rau 1 lub hlis ntawm 2-8℃nyob rau hauv kaw qhuav; nkoj ntawm cov pob khov nab kuab pom zoo. | Nyob ruaj khov rau 14 hnub ntawm 4 degree. Dawb soluble nyob rau hauv dej thiab physiological buffers. Disulfide daim ntawv cog lus yog rhiab rau cov muaj zog txo cov neeg ua haujlwm. Hauv vivo kev ruaj ntseg tom qab hloov kho yog qhov zoo dua li cov neeg vasopressin. | ruaj khov rau 3 xyoos ntawm -20 degree, qhuav thiab tiv thaiv los ntawm lub teeb. |
Functional Description
| Khoom Code | Frontend Short Summary (rau cov npe tshawb nrhiav) | Cov lus piav qhia txog kev ua haujlwm lom neeg lom neeg | Cov cheeb tsam tshawb fawb (comma- cais) | Lub Hom Phiaj / Txoj Kev |
| PEB-SEL001 | Tshiab- tiam tshiab xaiv V1a receptor agonist nrog cov nyhuv pressor thiab tsis muaj dej pom tseeb -sodium retention | Selepessin yog ib tug tshiab - tiam neeg xaiv vasopressin V1a receptor agonist. Nws tshwj xeeb khi rau V1a receptors ntawm vascular du leeg, muaj zog constricts peripheral resistance hlab ntsha thiab ua rau kom cov hlab ntsha siab, siv rau kev tshawb fawb kev kho mob hauv vasodilatory shock. Optimized los ntawm ntau yam -site amino acid ib ntus, nws tau txhim kho kev xaiv zoo rau V1a receptors thiab NW nyuam qhuav qhib V2 receptors, zam cov kev mob tshwm sim ntawm ib txwm muaj vasopressin xws li dej-sodium retention, antidiuresis thiab hyponatremia, nrog rau cov txiaj ntsig zoo dua thiab muaj kev nyab xeeb dua. Nws yog ib qho tshiab - tiam cuab tam peptide rau septic shock, vasodilatory hypotension, cardiovascular pharmacology thiab vasopressin receptor subtype kev tshawb fawb. | Septic/vasodilatory shock research, cardiovascular pharmacology study, vasopressin receptor subtype function research, pressor drug development, kev tshawb fawb hemodynamic | Vasopressin 1a receptor (V1aR); Vascular smooth nqaij contraction thiab ntshav siab tswj txoj kev |
Cim npe nrov: Tuam Tshoj selepessin acetate manufacturers, lwm tus neeg, Hoobkas
